Ubume bemolekyuli:
I-Cytisine yi-alkaloid eyenzeka ngokwemvelo efumaneka kwiintlobo ezininzi zezityalo, ezifana neCytisus laborinum kunye neLaburnum anagyroides. Isetyenziswe iminyaka emininzi njengoncedo lokuyeka ukutshaya ngenxa yokufana kwayo ne-nicotine.Umsebenzi oyintloko we-cytisine ufana ne-agonist inxalenye ye-nicotinic acetylcholine receptors (nAChRs). Ezi zamkeli zifunyanwa kwingqondo, ngokukodwa kwiindawo ezibandakanyekayo ekukhobokeni, kwaye zinoxanduva lokulamla iziphumo ezinomvuzo ze-nicotine. Ngokuzibophelela kunye nokusebenza kwezi receptors, i-cytisine inceda ekunciphiseni iminqweno ye-nicotine kunye neempawu zokurhoxisa ngexesha lokuyeka ukutshaya.I-Cytisine ibonakaliswe ukuba yonyango olusebenzayo lwe-nicotine umlutha kwizifundo ezahlukeneyo zeklinikhi. Inokukunceda ukuphucula amazinga okuyeka kunye nokunciphisa ubunzima beempawu zokurhoxisa, okwenza kube luncedo oluncedo kwiiprogram zokuyeka ukutshaya.
Kubalulekile ukuqaphela ukuba i-cytisine ingaba nemiphumo emibi, efana ne-nausea, ukuhlanza, kunye nokuphazamiseka kokulala. Njengalo naliphi na iyeza, kufuneka lisetyenziswe njengoko kuyalelwe kwaye phantsi kweliso lengcali yezempilo. Ukuba ucinga ukusebenzisa i-cytisine njengoncedo lokuyeka ukutshaya, ndincoma ukubonisana nogqirha wakho ngeengcebiso kunye nesikhokelo.
| Into | Inkcazo | |
| Uvavanyo (HPLC) | ||
| Cytisine: | ≥98% | |
| Umgangatho: | CP2010 | |
| Physicochemical | ||
| Imbonakalo: | Umgubo wekristale otyheli okhanyayo | |
| Ivumba: | uphawu oder | |
| Unizi lolwapho kuyiwa khona: | 50-60g/100ml | |
| Umnatha: | I-95% iphumelele i-80mesh | |
| Intsimbi enzima: | ≤10PPM | |
| Njengoko: | ≤2PPM | |
| Pb: | ≤2PPM | |
| Ilahleko yokomisa: | ≤1% | |
| Intsalela Ebasiweyo: | ≤0.1% | |
| Intsalela yokunyibilikisa: | ≤3000PPM | |