Isakhiwo samangqamuzana:
I-Cytisine iyi-alkaloid eyenzeka ngokwemvelo etholakala ezinhlobonhlobo zezitshalo ezimbalwa, njenge-Cytisus laborinum ne-Laburnum anagyroides. Isetshenziswe iminyaka eminingi njengosizo lokuyeka ukubhema ngenxa yokufana kwayo ne-nicotine.Umsebenzi oyinhloko we-cytisine ufana ne-agonist eyingxenye ye-nicotinic acetylcholine receptors (nAChRs). Lawa ma-receptors atholakala ebuchosheni, ikakhulukazi ezindaweni ezibandakanyeka ekuluthweni, futhi anesibopho sokulamula imiphumela enomvuzo ye-nicotine. Ngokubophezela nokusebenzisa lawa ma-receptors, i-cytisine isiza ukunciphisa izifiso ze-nicotine kanye nezimpawu zokuhoxiswa ngesikhathi sokuyeka ukubhema.I-Cytisine iboniswe njengendlela yokwelapha ephumelelayo yokulutha kwe-nicotine ezifundweni ezihlukahlukene zomtholampilo. Kungasiza ukuthuthukisa amazinga okuyeka futhi kunciphise ubukhali bezimpawu zokuhoxa, kukwenze kube usizo oluwusizo ezinhlelweni zokuyeka ukubhema.
Kubalulekile ukuqaphela ukuthi i-cytisine ingaba nemiphumela engemihle, njengokucanuzela kwenhliziyo, ukuhlanza, nokuphazamiseka kokulala. Njenganoma yimuphi umuthi, kufanele usetshenziswe njengoba kuyaliwe futhi ngaphansi kokugadwa uchwepheshe wezokunakekelwa kwempilo. Uma ucabanga ukusebenzisa i-cytisine njengosizo lokuyeka ukubhema, ngincoma ukuthi uxhumane nodokotela wakho ukuze uthole iseluleko esiqondene nawe kanye nesiqondiso.
| Into | Ukucaciswa | |
| I-Assay (HPLC) | ||
| I-Cytisine: | ≥98% | |
| Okujwayelekile: | I-CP2010 | |
| I-Physicochemical | ||
| Ukubukeka: | Impushana yekristalu ephuzi ekhanyayo | |
| Iphunga: | I-oda yesici | |
| Ukuminyana kwenqwaba: | 50-60g/100ml | |
| I-Mesh: | U-95% uphase ama-80mesh | |
| Insimbi enzima: | ≤10PPM | |
| Njengo: | ≤2PPM | |
| I-Pb: | ≤2PPM | |
| Ukulahlekelwa Kokomisa: | ≤1% | |
| Izinsalela Ezibasiwe: | ≤0.1% | |
| I-Solvent Residue: | ≤3000PPM | |